4e5d A 2.201 BS01 0NJ A 1 H245 G246 F247 G315 G341 L342 T343 S347 A348 H238 G239 F240 G308 G331 L332 T333 S337 A338 S198 R218 H245 T343 E344 S196 R211 H238 T333 E334 1.13.12.7 0001676,0004467,0004497,0005524,0005777,0008218,0046872,0046949,0047077,0051087 -logKd/Ki=6.22, IC50=0.6uM IC50=600nM P08659 22921073 601 DAKNIKKGPAPFYPLEDGTAGEQLHKAMKRYALVPGTIAFTDAHIEVNITYAEYFEMSVRLAEAMKRYGLNTNHRIVVCSENSLQFFMPVLGALFIGVAVAPANDIYNERELLNSMNISQPTVVFVSKKGLQKILNVQKKLPIIQKIIIMDSKTDYQGFQSMYTFVTSHLPPGFNEYDFVPESFDRDKTIALIMNSLPKGVALPHRTACVRFSHARDPIFGNQIIPDTAILSVVPFHHGFGMFTTLGYLICGFRVVLMYRFEEELFLRSLQDYKIQSALLVPTLFSFFAKSTLIDKYDLSNLHEIASGLSKEVGEAVAKRFHLPGIRQGYGLTETTSAILITPEGDDKPGAVGKVVPFFEAKVVDLDTGKTLGVNQRGELCVRGPMIMSGYVNNPEATNALIDKDGWLHSGDIAYWDEDEHFFIV