4e0x A 2.0 BS01 KAI A 1 E13 Y61 P88 T90 R95 G140 S141 T142 E190 E10 Y58 P85 T87 R92 G137 S138 T139 E187 ? 0015276,0016020 -logKd/Ki=7.12, Ki=76nM IC50=77nM, Ki=75.9nM, EC50=37000nM P22756 22425692 301 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWR 4e0x B 2.0 BS01 KAI B 1 E13 Y61 P88 T90 R95 G140 S141 T142 E190 E10 Y58 P85 T87 R92 G137 S138 T139 E187 ? 0015276,0016020 IC50=77nM, Ki=75.9nM, EC50=37000nM P22756 22425692 301 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP