4deg A 2.0 BS01 0JJ A 1 I1084 A1108 M1160 D1164 R1208 M1211 A1221 D1222 Y1230 I33 A51 M100 D104 R148 M151 A161 D162 Y170 D1204 A1206 R1208 N1209 D1222 A1243 D144 A146 R148 N149 D162 A183 2.7.10.1 0004672,0004713,0005524,0006468 ic50=6nM -logKd/Ki=8.22, IC50=6nM IC50=3nM, Ki=3.2nM P08581 22595176 1401 HIDLSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLKIHCAVKSLNRITDIGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIG