4ded A 3.05 BS01 NHU A 1 R137 L139 G140 V147 A160 K162 A213 G216 R220 L263 R14 L16 G17 V24 A37 K39 A90 G93 R97 L140 D256 K258 E260 N261 D274 T292 D133 K135 E137 N138 D151 T169 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=7.42, IC50=38.2nM IC50=38.2nM O14965 22803810 501 KKRQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRDTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS