4btt B 2.59 BS01 CA B 1 D70 N72 Q75 E77 E80 D56 N58 Q61 E63 E66 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 P00742 24175584 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4btt B 2.59 BS02 VYR B 1 H57 Q61 Y99 F174 A190 Q192 V213 S214 W215 G216 G226 Y228 H42 Q46 Y85 F162 A180 Q182 V203 S204 W205 G206 G216 Y218 H57 D102 Q192 G193 D194 S195 G196 H42 D88 Q182 G183 D184 S185 G186 3.4.21.6 0004252,0006508 IC50=2.6nM P00742 24175584 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4btt F 2.59 BS01 CA F 1 D70 N72 Q75 E76 E80 D56 N58 Q61 E62 E66 G193 S195 G196 G183 S185 G186 3.4.21.6 0004252,0006508 P00742 24175584 1245 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT 4btt F 2.59 BS02 VYR F 1 Q61 T98 Y99 F174 A190 Q192 V213 S214 W215 G216 G226 Y228 Q46 T84 Y85 F162 A180 Q182 V203 S204 W205 G206 G216 Y218 G193 S195 G196 G183 S185 G186 3.4.21.6 0004252,0006508 -logKd/Ki=8.84, IC50=1.43nM IC50=2.6nM P00742 24175584 1246 IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRFTKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSSSFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT