4bdo A 2.55 BS01 KAI A 1 E440 Y488 P516 A518 R523 G688 A689 T690 E738 E10 Y54 P78 A80 R85 G130 A131 T132 E180 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 RSLIVTTILEEPYVLFKKLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKIGIAILQLQEEGKLHMMKEKWWR 4bdo B 2.55 BS01 KAI B 1 E440 Y488 P516 A518 R523 G688 A689 T690 E738 E9 Y52 P80 A82 R87 G132 A133 T134 E182 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 SLIVTTILEEPYVLFKLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKIGIAILQLQEEGKLHMMKEKWWRC 4bdo C 2.55 BS01 KAI C 1 E440 Y488 P516 L517 A518 R523 G688 A689 T690 E738 E9 Y54 P82 L83 A84 R89 G134 A135 T136 E184 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 SLIVTTILEEPYVLFKKSLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKIGIAILQLQEEGKLHMMKEKWWR 4bdo D 2.55 BS01 KAI D 1 E440 Y488 P516 A518 R523 G688 A689 T690 E738 E9 Y52 P75 A77 R82 G127 A128 T129 E177 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 SLIVTTILEEPYVLFKLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKIGIAILQLQEEGKLHMMKEKWWRC 4bdo D 2.55 BS02 GLU D 1 Y488 L517 A518 R523 G688 A689 T690 E738 Y52 L76 A77 R82 G127 A128 T129 E177 ? 0015276,0016020 P42260 23720540 901 SLIVTTILEEPYVLFKLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKIGIAILQLQEEGKLHMMKEKWWRC