4bdm A 3.4 BS01 KAI A 1 Y488 P516 A518 R523 V685 G688 A689 T690 E738 Y57 P83 A85 R90 V132 G135 A136 T137 E185 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWW 4bdm B 3.4 BS01 KAI B 1 E440 Y488 P516 A518 R523 V685 G688 A689 T690 E738 E9 Y57 P85 A87 R92 V134 G137 A138 T139 E187 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWW 4bdm C 3.4 BS01 KAI C 1 E440 Y488 P516 L517 A518 R523 G688 A689 T690 E738 E9 Y57 P85 L86 A87 R92 G137 A138 T139 E187 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWW 4bdm D 3.4 BS01 KAI D 1 Y488 P516 A518 R523 G688 A689 T690 E738 Y57 P85 A87 R92 G137 A138 T139 E187 ? 0015276,0016020 Ki=12.7nM, Kd=39nM, EC50=1800nM P42260 23720540 900 SLIVTTILEEPYVLFKKSDKPLYGNDRFEGYCIDLLRELSTILGFTYEIRLVEDGKYGAQDDVNGQWNGMVRELIDHKADLAVAPLAITYVREKVIDFSAPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVEDGATMTFFKKSKISTYDKMWAFMSSRRQSVLVKSNEEGIQRVLTSDYAFLMESTTIEFVTQRNCNLTQIGGLIDSKGYGVGTPMGSPYRDKITIAILQLQEEGKLHMMKEKWW