4awg A 2.6 BS01 CI3 A 1 E23 Y24 A37 I38 H41 E80 R84 D108 E119 K134 E26 Y27 A40 I41 H44 E77 R81 D105 E116 K131 3.1.-.- 0003723,0039694 -logKd/Ki=5.96, IC50=1.1uM C3W5S0 22876177 801 GMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVELLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQS 4awg A 2.6 BS02 MN A 1 H41 D108 E119 I120 H44 D105 E116 I117 3.1.-.- 0003723,0039694 C3W5S0 22876177 901 GMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVELLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQS 4awg A 2.6 BS03 MN A 2 E80 D108 E77 D105 3.1.-.- 0003723,0039694 C3W5S0 22876177 902 GMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVELLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQS 4awg B 2.6 BS01 CI3 B 1 E23 Y24 K34 A37 I38 H41 R84 D108 E119 K134 E26 Y27 K37 A40 I41 H44 R81 D105 E116 K131 3.1.-.- 0003723,0039694 C3W5S0 22876177 801 GMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVELLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQS 4awg B 2.6 BS02 MN B 1 H41 D108 E119 I120 H44 D105 E116 I117 3.1.-.- 0003723,0039694 C3W5S0 22876177 901 GMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVELLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQS 4awg B 2.6 BS03 MN B 2 E80 D108 E77 D105 3.1.-.- 0003723,0039694 C3W5S0 22876177 902 GMAMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVELLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQS 4awg C 2.6 BS01 CI3 C 1 A20 E23 Y24 I38 H41 E80 D108 E119 K134 A21 E24 Y25 I39 H42 E81 D109 E120 K135 3.1.-.- 0003723,0039694 C3W5S0 22876177 801 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4awg C 2.6 BS02 MN C 1 H41 D108 E119 I120 H42 D109 E120 I121 3.1.-.- 0003723,0039694 C3W5S0 22876177 901 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4awg C 2.6 BS03 MN C 2 E80 D108 E81 D109 3.1.-.- 0003723,0039694 C3W5S0 22876177 902 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFHFIDERGESIIVESGDPNALLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4awg D 2.6 BS01 CI3 D 1 E23 Y24 I38 H41 E80 R84 D108 E119 K134 E24 Y25 I39 H42 E61 R65 D89 E100 K115 3.1.-.- 0003723,0039694 C3W5S0 22876177 801 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4awg D 2.6 BS02 MN D 1 H41 D108 E119 I120 H42 D89 E100 I101 3.1.-.- 0003723,0039694 C3W5S0 22876177 901 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE 4awg D 2.6 BS03 MN D 2 E80 D108 E61 D89 3.1.-.- 0003723,0039694 C3W5S0 22876177 902 AMEDFVRQCFNPMIVELAEKAMKEYGEDPKIETNKFAAICTHLEVCFMYSDFLKHRFEIIEGRDRIMAWTVVNSICNTTGVEKPKFLPDLYDYKENRFIEIGVTRREVHIYYLEKANKIKSEKTHIHIFSFTGEEMATKADYTLDEESRARIKTRLFTIRQEMASRSLWDSFRQSE