4asy A 2.3 BS01 N5Y A 1 S41 T42 L45 Y113 G115 V250 E255 S41 T42 L45 Y113 G115 V250 E255 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 -logKd/Ki=4.22, IC50>60uM IC50=>6.0e+4nM Q9HU22 23138692 1294 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4asy B 2.3 BS01 N5Y B 1 S41 L45 Y113 G115 V250 E255 S40 L44 Y112 G114 V249 E254 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 -logKd/Ki=4.22, IC50>60uM IC50=>6.0e+4nM Q9HU22 23138692 1294 KRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4asy C 2.3 BS01 N5Y C 1 S41 L45 Y113 Y114 G115 V250 E255 S41 L45 Y113 Y114 G115 V250 E255 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 IC50=>6.0e+4nM Q9HU22 23138692 1294 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY 4asy D 2.3 BS01 N5Y D 1 S41 L45 Y113 Y114 G115 E255 Q260 S41 L45 Y113 Y114 G115 E255 Q260 2.7.7.24 0000166,0008879,0009058,0009244,0016779,0019305,0045226,0046872 IC50=>6.0e+4nM Q9HU22 23138692 1294 MKRKGIILAGGSGTRLHPATLAISKQLLPVYDKPMIYYPLSTLMLAGIREILIISTPQDTPRFQQLLGDGSNWGLDLQYAVQPSPDGLAQAFLIGESFIGNDLSALVLGDNLYYGHDFHELLGSASQRQTGASVFAYHVLDPERYGVVEFDQGGKAISLEEKPLEPKSNYAVTGLYFYDQQVVDIARDLKPSPRGELEITDVNRAYLERGQLSVEIMGRGYAWLDTGTHDSLLEAGQFIATLENRQGLKVACPEEIAYRQKWIDAAQLEKLAAPLAKNGYGQYLKRLLTETVY