4an9	A	2.8	BS01	ACP	A	1	L74 G75 A76 G77 N78 A95 M143 M146 Q153 K192 S194 L197	L17 G18 A19 G20 N21 A38 M86 M89 Q96 K135 S137 L140	D190 K192 S194 N195 D208 D217 T226	D133 K135 S137 N138 D151 D160 T168	2.7.12.2	0004672,0005524,0006468					Q02750	24900486	1382 	MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL
4an9	A	2.8	BS02	MG	A	1	N195 D208	N138 D151	D190 K192 S194 N195 D208 D217 T226	D133 K135 S137 N138 D151 D160 T168	2.7.12.2	0004672,0005524,0006468					Q02750	24900486	1383 	MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL
4an9	A	2.8	BS03	2P7	A	1	K97 L118 V127 I141 M143 D190 D208 F209 G210 V211 L215	K40 L61 V70 I84 M86 D133 D151 F152 G153 V154 L158	D190 K192 S194 N195 D208 D217 T226	D133 K135 S137 N138 D151 D160 T168	2.7.12.2	0004672,0005524,0006468			-logKd/Ki=7.36, IC50=44nM	IC50=44nM	Q02750	24900486	1384 	MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL