4aig A 2.0 BS01 ZN A 1 H142 H146 H152 H141 H145 H151 3.4.24.46 0004222,0005576,0005886,0006508,0008237,0046872 P34179 9428736 999 NLPQRYIELVVVADRRVFMKYNSDLNIIRTRVHEIVNIINEFYRSLNIRVSLTDLEIWSGQDFITIQSSSSNTLNSFGEWRERVLLTRKRHDNAQLLTAINFEGKIIGKAYTSSMCNPRSSVGIVKDHSPINLLVAVTMAHELGHNLGMEHDGKDCLRGASLCIMRPGLTPGRSYEFSDDSMGYYQKFLNQYKPQCILNKP 4aig A 2.0 BS02 CA A 1 E9 D93 C197 N200 E8 D92 C196 N199 3.4.24.46 0004222,0005576,0005886,0006508,0008237,0046872 P34179 9428736 250 NLPQRYIELVVVADRRVFMKYNSDLNIIRTRVHEIVNIINEFYRSLNIRVSLTDLEIWSGQDFITIQSSSSNTLNSFGEWRERVLLTRKRHDNAQLLTAINFEGKIIGKAYTSSMCNPRSSVGIVKDHSPINLLVAVTMAHELGHNLGMEHDGKDCLRGASLCIMRPGLTPGRSYEFSDDSMGYYQKFLNQYKPQCILNKP 4aig A 2.0 BS03 FLX A 1 K106 I107 I108 T139 H142 E143 H146 H152 I165 R167 P168 G169 L170 K105 I106 I107 T138 H141 E142 H145 H151 I164 R166 P167 G168 L169 3.4.24.46 0004222,0005576,0005886,0006508,0008237,0046872 ic50=0.3uM -logKd/Ki=6.52, IC50=0.3uM P34179 9428736 400 NLPQRYIELVVVADRRVFMKYNSDLNIIRTRVHEIVNIINEFYRSLNIRVSLTDLEIWSGQDFITIQSSSSNTLNSFGEWRERVLLTRKRHDNAQLLTAINFEGKIIGKAYTSSMCNPRSSVGIVKDHSPINLLVAVTMAHELGHNLGMEHDGKDCLRGASLCIMRPGLTPGRSYEFSDDSMGYYQKFLNQYKPQCILNKP