3zc6 A 2.42 BS01 VFC A 1 L828 G829 K830 G831 G834 V836 A853 K855 E903 Y904 L905 G908 C909 L956 D967 L15 G16 K17 G18 G21 V23 A40 K42 E86 Y87 L88 G91 C92 L139 D150 D949 A951 R953 N954 D967 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM -logKd/Ki=9.22, IC50=0.6nM IC50=0.600000nM P52333 23540648 2103 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 3zc6 B 2.42 BS01 VFC B 1 L828 G829 K830 G831 G834 V836 A853 K855 M902 E903 Y904 L905 G908 L956 L16 G17 K18 G19 G22 V24 A41 K43 M86 E87 Y88 L89 G92 L140 D949 A951 R953 N954 D967 D133 A135 R137 N138 D151 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM IC50=0.600000nM P52333 23540648 2103 DPTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 3zc6 C 2.42 BS01 VFC C 1 L828 G829 K830 G831 G834 V836 A853 K855 M902 E903 Y904 L905 G908 C909 L956 D967 L15 G16 K17 G18 G21 V23 A40 K42 M83 E84 Y85 L86 G89 C90 L137 D148 D949 A951 R953 N954 D967 D130 A132 R134 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM IC50=0.600000nM P52333 23540648 2103 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVRSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGSERDVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS 3zc6 D 2.42 BS01 VFC D 1 L828 G829 K830 G831 G834 S835 V836 A853 K855 M902 E903 Y904 L905 G908 L956 L15 G16 K17 G18 G21 S22 V23 A40 K42 M84 E85 Y86 L87 G90 L138 D949 A951 R953 N954 D967 D131 A133 R135 N136 D149 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM IC50=0.600000nM P52333 23540648 2103 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVRPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMLSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWS