3wzk A 2.3 BS01 O23 A 1 I531 Q541 K553 E571 M602 C604 G605 N606 L654 I663 I16 Q26 K38 E56 M87 C89 G90 N91 L139 I148 D647 K649 N652 D664 D674 T686 D132 K134 N137 D149 D159 T161 2.7.12.1 0004672,0005524,0006468 ic50=58nM -logKd/Ki=7.24, IC50=58nM IC50=561nM P33981 25625617 901 ECISVKGRIYSILKQIGSGGSSKVFQVLNEKKQIYAIKYVNLEEADNQTLDSYRNEIAYLNKLQQHSDKIIRLYDYEITDQYIYMVMECGNIDLNSWLKKKKSIDPWERKSYWKNMLEAVHTIHQHGIVHSDLKPANFLIVDGMLKLIDFGIANQMQPDGTVNYMPPEAIKDMSISPKSDVWSLGCILYYMTYGKTPFQQIINQISKLHAIIDPNHEIEFPDIPEKDLQDVLKCCLKRDPKQRISIPELLAHPYVQIQ