3w4j A 2.74 BS01 FAD A 1 G7 A8 G9 V10 I11 A36 D37 R38 T44 T45 A48 G50 L51 V164 T182 W185 G312 G313 Y314 G315 L316 T317 G7 A8 G9 V10 I11 A36 D37 R38 T44 T45 A48 G50 L51 V164 T182 W185 G312 G313 Y314 G315 L316 T317 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 P14920 23566269 401 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS 3w4j A 2.74 BS02 2LD A 1 Q53 L215 H217 Y224 Y228 R283 G313 Q53 L215 H217 Y224 Y228 R283 G313 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 IC50=20nM P14920 23566269 402 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS 3w4j B 2.74 BS01 FAD B 1 I6 G7 G9 V10 I11 A36 D37 R38 T44 T45 A48 G50 L51 V164 T182 R283 G312 G313 Y314 G315 L316 T317 I6 G7 G9 V10 I11 A36 D37 R38 T44 T45 A48 G50 L51 V164 T182 R283 G312 G313 Y314 G315 L316 T317 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 P14920 23566269 401 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS 3w4j B 2.74 BS02 2LD B 1 Q53 Y224 Y228 R283 G313 Q53 Y224 Y228 R283 G313 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 IC50=20nM P14920 23566269 402 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS 3w4j C 2.74 BS01 FAD C 1 G7 A8 G9 V10 I11 A36 D37 R38 T44 T45 A48 G50 L51 K163 V164 T182 R283 G312 G313 Y314 G315 L316 T317 G7 A8 G9 V10 I11 A36 D37 R38 T44 T45 A48 G50 L51 K163 V164 T182 R283 G312 G313 Y314 G315 L316 T317 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 P14920 23566269 401 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS 3w4j C 2.74 BS02 2LD C 1 Q53 L215 H217 Y224 Y228 I230 R283 G313 Q53 L215 H217 Y224 Y228 I230 R283 G313 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 IC50=20nM P14920 23566269 402 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS 3w4j D 2.74 BS01 FAD D 1 G7 A8 G9 I11 A36 D37 R38 T43 T44 T45 A48 G50 L51 R162 K163 V164 T182 W185 G313 G315 L316 T317 G7 A8 G9 I11 A36 D37 R38 T43 T44 T45 A48 G50 L51 R162 K163 V164 T182 W185 G313 G315 L316 T317 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 P14920 23566269 401 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS 3w4j D 2.74 BS02 2LD D 1 Q53 L215 H217 Y224 Y228 R283 G313 Q53 L215 H217 Y224 Y228 R283 G313 L51 G313 T317 L51 G313 T317 1.4.3.3 0003884,0005515,0005576,0005737,0005741,0005777,0005782,0005829,0006562,0007586,0016491,0019478,0036088,0042416,0042802,0042995,0045202,0046416,0048786,0055130,0070178,0070945,0071949 IC50=20nM P14920 23566269 402 MRVVVIGAGVIGLSTALCIHERYHSVLQPLDIKVYADRFTPLTTTDVAAGLWQPYLSDPNNPQEADWSQQTFDYLLSHVHSPNAENLGLFLISGYNLFHEAIPDPSWKDTVLGFRKLTPRELDMFPDYGYGWFHTSLILEGKNYLQWLTERLTERGVKFFQRKVESFEEVAREGADVIVNCTGVWAGALQRDPLLQPGRGQIMKVDAPWMKHFILTHDPERGIYNSPYIIPGTQTVTLGGIFQLGNWSELNNIQDHNTIWEGCCRLEPTLKNARIIGERTGFRPVRPQIRLEREQLRTGPSNTEVIHNYGHGGYGLTIHWGCALEAAKLFGRILEEKKLS