3vf8 A 2.08 BS01 0JE A 1 L377 A400 M450 A451 E452 G454 P455 L501 S511 L15 A36 M80 A81 E82 G84 P85 L131 S141 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K163 2.7.10.2 0004672,0004713,0005524,0006468 ic50=150nM -logKd/Ki=6.82, IC50=150nM P43405 22464456 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN