3tjc A 2.4 BS01 0TP A 1 L855 G856 Y931 L932 G935 N981 L983 D994 L13 G14 Y85 L86 G89 N135 L137 D148 D976 A978 R980 N981 D994 S1016 D130 A132 R134 N135 D148 S170 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.031uM -logKd/Ki=7.51, IC50=31nM IC50=3940nM O60674 22087750 1 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 3tjc B 2.4 BS01 0TP B 1 L855 G858 V863 Y931 L932 P933 G935 L983 L16 G19 V24 Y88 L89 P90 G92 L140 D976 A978 R980 N981 D994 S1016 D133 A135 R137 N138 D151 S173 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.031uM IC50=3940nM O60674 22087750 1 DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG