3t8s B 3.77 BS01 I3P B 1 R265 T267 Y567 R568 R251 T253 Y469 R470 ? 0005220,0005262,0005783,0006816,0016020,0070588,0070679 -logKd/Ki=8.55, Kd=2.82nM Kd=8.7nM, EC50=209nM P29994 21892169 603 SFLHIGDICSLYAEGSTNGFISTLGLVDDRCVVQPEAGDLNNPPKKFRDCLFKLCPMNRYSAQKQFWKTTDAVLLNKLHHAADLEKKQNETENRKLLGTVIQYGNVIQLLHLKSNKYLTVNKRLPALLEKNAMRVTLDEAGNEGSWFYIQPFYKLRSIGDSVVIGDKVVLNPVNAGQPLHASSHQLVDNPGCNEVNSVNCNTSWKIVLFMKWSDNKDDILKGGDVVRLFHAEQEKFLTCDEHRKKQHVFLRTTSATSSKALWEVEVVQHDPWNSLFRFKHLATGHYLAAEVDYSLVSVPEGNDISSIFELDPLVPRNSYVRLRHLCTNTWVHSTNIPIDKEEEKPVMLKIGTSPLKEDKEAFAIVPVSPAEVRDLDFANDASKVLGSIAGKLEKGTITQNERRSVTKLLEDLVYFVTGEVVFSKPNRERQKLMREQNILKQIFKLLQAPPFRHICRLCYRVLRHSQQDYRKNQEYIAKQFGF