3sfi A 2.31 BS01 3SF A 1 M102 G106 F110 F114 W138 W145 Y148 T149 N176 N179 E180 W207 M81 G85 F89 F93 W117 W124 Y127 T128 N155 N158 E159 W186 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.4uM -logKd/Ki=6.40, IC50=0.4uM IC50=400nM, EC50=60nM P9WMC1 22098589 217 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGE