3ro0 A 1.5 BS01 TPT A 1 F10 F13 N19 T45 A139 F142 C144 H168 F9 F12 N18 T44 A138 F141 C143 H167 E81 R91 C144 H168 E80 R90 C143 H167 3.4.19.3 0005737,0005829,0006508,0008234,0016920 -logKd/Ki=4.50, IC50=31.89uM P46107 21875148 480 EKKVLLTGFDPFGGETVNPSWEAVKRLNGAAEGPASIVSEQVPTVFYKSLAVLREAMKKHQPDIIICVGQAGGRMQITPERVAINLNEARIPDNEGNQPVGEDISQGGPAAYWTGLPIKRIVEEIKKEGIPAAVSYTAGTFVCNHLFYGLMDEISRHHPHIRGGFIHIPYIPEQTLQKSAPSLSLDHITKALKIAAVTAAAHEDDIE 3ro0 B 1.5 BS01 TPT B 1 F10 F13 T45 A139 C144 H168 F10 F13 T45 A139 C144 H168 E81 R91 C144 H168 E81 R91 C144 H168 3.4.19.3 0005737,0005829,0006508,0008234,0016920 P46107 21875148 481 MEKKVLLTGFDPFGGETVNPSWEAVKRLNGAAEGPASIVSEQVPTVFYKSLAVLREAMKKHQPDIIICVGQAGGRMQITPERVAINLNEARIPDNEGNQPVGEDISQGGPAAYWTGLPIKRIVEEIKKEGIPAAVSYTAGTFVCNHLFYGLMDEISRHHPHIRGGFIHIPYIPEQTLQKSAPSLSLDHITKALKIAAVTAAAHEDDIET 3ro0 C 1.5 BS01 TPT C 1 F10 F13 T45 A139 F142 C144 H168 F10 F13 T45 A139 F142 C144 H168 E81 R91 C144 H168 E81 R91 C144 H168 3.4.19.3 0005737,0005829,0006508,0008234,0016920 P46107 21875148 482 MEKKVLLTGFDPFGGETVNPSWEAVKRLNGAAEGPASIVSEQVPTVFYKSLAVLREAMKKHQPDIIICVGQAGGRMQITPERVAINLNEARIPDNEGNQPVGEDISQGGPAAYWTGLPIKRIVEEIKKEGIPAAVSYTAGTFVCNHLFYGLMDEISRHHPHIRGGFIHIPYIPEQTLQKSAPSLSLDHITKALKIAAVTAAAHEDDI 3ro0 D 1.5 BS01 TPT D 1 F10 F13 T45 A139 F142 C144 H168 F9 F12 T44 A138 F141 C143 H167 E81 R91 C144 H168 E80 R90 C143 H167 3.4.19.3 0005737,0005829,0006508,0008234,0016920 P46107 21875148 483 EKKVLLTGFDPFGGETVNPSWEAVKRLNGAAEGPASIVSEQVPTVFYKSLAVLREAMKKHQPDIIICVGQAGGRMQITPERVAINLNEARIPDNEGNQPVGEDISQGGPAAYWTGLPIKRIVEEIKKEGIPAAVSYTAGTFVCNHLFYGLMDEISRHHPHIRGGFIHIPYIPEQTLQKSAPSLSLDHITKALKIAAVTAAAHEDDI 3ro0 D 1.5 BS02 TPT D 2 H158 H159 P160 H161 H157 H158 P159 H160 E81 R91 C144 H168 E80 R90 C143 H167 3.4.19.3 0005737,0005829,0006508,0008234,0016920 P46107 21875148 484 EKKVLLTGFDPFGGETVNPSWEAVKRLNGAAEGPASIVSEQVPTVFYKSLAVLREAMKKHQPDIIICVGQAGGRMQITPERVAINLNEARIPDNEGNQPVGEDISQGGPAAYWTGLPIKRIVEEIKKEGIPAAVSYTAGTFVCNHLFYGLMDEISRHHPHIRGGFIHIPYIPEQTLQKSAPSLSLDHITKALKIAAVTAAAHEDDI