3rhq A 2.1 BS01 NAP A 1 V570 I571 P572 W573 N574 K597 A599 Q600 S629 G630 G634 Q635 F648 T649 G650 S651 V654 I658 E673 L674 A707 E804 F806 V166 I167 P168 W169 N170 K193 A195 Q196 S225 G226 G230 Q231 F244 T245 G246 S247 V250 I254 E269 L270 A303 E400 F402 N574 K597 E673 A707 E804 D883 N170 K193 E269 A303 E400 D479 1.5.1.6 0016491,0016620 Kd=9.2uM P28037 21540484 903 VINYVEKAVNKLTLQMPYQLFIGGEFVDAEGSKTYNTINPTDGSVICQVSLAQVSDVDKAVAAAKEAFENGLWGKINARDRGRLLYRLADVMEQHQEELATIEALDAGAVYTLALKTHVGMSIQTFRYFAGWCDKIQGATIPINQARPNRNLTLTKKEPVGVCGIVIPWNYPLMMLSWKTAACLAAGNTVVIKPAQVTPLTALKFAELTLKAGIPKGVVNILPGSGSLVGQRLSDHPDVRKIGFTGSTEVGKHIMKSCALSNVKKVSLELGGKSPLIIFADCDLNKAVQMGMSSVFFNKGENAIAAGRLFVEESIHNQFVQKVVEEVEKMKIGNPLERDTNHGPQNHEAHLRKLVEYCQRGVKEGATLVCGGNQVPRPGFFFQPTVFTDVEDHMYIAKEESFGPIMIISRFADGDVDAVLSRANATEFGLASGVFTRDINKALYVSDKLQAGTVFINTYNKTDVAAPFGGFKQSGFGKDLGEAALNEYLRIKTVTFEY 3rhq B 2.1 BS01 NAP B 1 V570 I571 P572 W573 N574 K597 A599 Q600 S629 G630 G634 Q635 F648 T649 G650 S651 V654 I658 E673 L674 G675 A707 E804 F806 F872 V166 I167 P168 W169 N170 K193 A195 Q196 S225 G226 G230 Q231 F244 T245 G246 S247 V250 I254 E269 L270 G271 A303 E400 F402 F468 N574 K597 E673 A707 E804 D883 N170 K193 E269 A303 E400 D479 1.5.1.6 0016491,0016620 Kd=9.2uM P28037 21540484 903 VINYVEKAVNKLTLQMPYQLFIGGEFVDAEGSKTYNTINPTDGSVICQVSLAQVSDVDKAVAAAKEAFENGLWGKINARDRGRLLYRLADVMEQHQEELATIEALDAGAVYTLALKTHVGMSIQTFRYFAGWCDKIQGATIPINQARPNRNLTLTKKEPVGVCGIVIPWNYPLMMLSWKTAACLAAGNTVVIKPAQVTPLTALKFAELTLKAGIPKGVVNILPGSGSLVGQRLSDHPDVRKIGFTGSTEVGKHIMKSCALSNVKKVSLELGGKSPLIIFADCDLNKAVQMGMSSVFFNKGENAIAAGRLFVEESIHNQFVQKVVEEVEKMKIGNPLERDTNHGPQNHEAHLRKLVEYCQRGVKEGATLVCGGNQVPRPGFFFQPTVFTDVEDHMYIAKEESFGPIMIISRFADGDVDAVLSRANATEFGLASGVFTRDINKALYVSDKLQAGTVFINTYNKTDVAAPFGGFKQSGFGKDLGEAALNEYLRIKTVTFEY 3rhq C 2.1 BS01 NAP C 1 V570 I571 P572 W573 N574 K597 A599 Q600 S629 G630 G634 Q635 F648 T649 G650 S651 V654 I658 E673 L674 A707 E804 F806 F872 V166 I167 P168 W169 N170 K193 A195 Q196 S225 G226 G230 Q231 F244 T245 G246 S247 V250 I254 E269 L270 A303 E400 F402 F468 N574 K597 E673 A707 E804 D883 N170 K193 E269 A303 E400 D479 1.5.1.6 0016491,0016620 Kd=9.2uM P28037 21540484 903 VINYVEKAVNKLTLQMPYQLFIGGEFVDAEGSKTYNTINPTDGSVICQVSLAQVSDVDKAVAAAKEAFENGLWGKINARDRGRLLYRLADVMEQHQEELATIEALDAGAVYTLALKTHVGMSIQTFRYFAGWCDKIQGATIPINQARPNRNLTLTKKEPVGVCGIVIPWNYPLMMLSWKTAACLAAGNTVVIKPAQVTPLTALKFAELTLKAGIPKGVVNILPGSGSLVGQRLSDHPDVRKIGFTGSTEVGKHIMKSCALSNVKKVSLELGGKSPLIIFADCDLNKAVQMGMSSVFFNKGENAIAAGRLFVEESIHNQFVQKVVEEVEKMKIGNPLERDTNHGPQNHEAHLRKLVEYCQRGVKEGATLVCGGNQVPRPGFFFQPTVFTDVEDHMYIAKEESFGPIMIISRFADGDVDAVLSRANATEFGLASGVFTRDINKALYVSDKLQAGTVFINTYNKTDVAAPFGGFKQSGFGKDLGEAALNEYLRIKTVTFEY 3rhq D 2.1 BS01 NAP D 1 V570 I571 P572 W573 N574 K597 A599 Q600 S629 G630 G634 Q635 F648 T649 G650 S651 V654 I658 E673 L674 G675 A707 E804 F806 V166 I167 P168 W169 N170 K193 A195 Q196 S225 G226 G230 Q231 F244 T245 G246 S247 V250 I254 E269 L270 G271 A303 E400 F402 N574 K597 E673 A707 E804 D883 N170 K193 E269 A303 E400 D479 1.5.1.6 0016491,0016620 Kd=9.2uM P28037 21540484 903 VINYVEKAVNKLTLQMPYQLFIGGEFVDAEGSKTYNTINPTDGSVICQVSLAQVSDVDKAVAAAKEAFENGLWGKINARDRGRLLYRLADVMEQHQEELATIEALDAGAVYTLALKTHVGMSIQTFRYFAGWCDKIQGATIPINQARPNRNLTLTKKEPVGVCGIVIPWNYPLMMLSWKTAACLAAGNTVVIKPAQVTPLTALKFAELTLKAGIPKGVVNILPGSGSLVGQRLSDHPDVRKIGFTGSTEVGKHIMKSCALSNVKKVSLELGGKSPLIIFADCDLNKAVQMGMSSVFFNKGENAIAAGRLFVEESIHNQFVQKVVEEVEKMKIGNPLERDTNHGPQNHEAHLRKLVEYCQRGVKEGATLVCGGNQVPRPGFFFQPTVFTDVEDHMYIAKEESFGPIMIISRFADGDVDAVLSRANATEFGLASGVFTRDINKALYVSDKLQAGTVFINTYNKTDVAAPFGGFKQSGFGKDLGEAALNEYLRIKTVTFEY