3rf4 A 1.8 BS01 FUN A 1 P1 M2 K32 R36 I64 V106 F108 V113 P1 M2 K32 R36 I64 V106 F108 V113 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=0.56uM -logKd/Ki=6.25, Ki=0.56uM A4GRE3 21944748 201 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf4 A 1.8 BS02 ZN A 1 E20 D24 E20 D24 ? 0005125,0005126,0005615,0007165,0046872,0050178 A4GRE3 21944748 119 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf4 B 1.8 BS01 FUN B 1 P1 M2 K32 R36 I64 V106 F108 P1 M2 K32 R36 I64 V106 F108 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=0.56uM A4GRE3 21944748 202 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf4 B 1.8 BS02 ZN B 1 E20 D24 E20 D24 ? 0005125,0005126,0005615,0007165,0046872,0050178 A4GRE3 21944748 120 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf4 B 1.8 BS03 FUN C 1 H49 I95 H49 I95 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=0.56uM A4GRE3 21944748 203 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA 3rf4 C 1.8 BS01 FUN C 1 P1 M2 K32 R36 I64 V106 F108 V113 P1 M2 K32 R36 I64 V106 F108 V113 ? 0005125,0005126,0005615,0007165,0046872,0050178 Ki=0.56uM -logKd/Ki=6.25, Ki=0.56uM A4GRE3 21944748 203 PMVRVATNLPDKDVPANFEERLTDLLAESMNKPRNRIAIEVLAGQRITHGASRNPVAVIKVESIGALSADDNIRHTQKITQFCQDTLKLPKDKVIITYFDLQPIHVGFNGTTVAAA