3pa3 A 1.4 BS01 C70 A 1 L15 A36 E85 Y86 C87 G90 E134 N135 L137 D148 K271 L11 A32 E73 Y74 C75 G78 E122 N123 L125 D136 K259 D130 K132 E134 N135 D148 T170 D118 K120 E122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1nM -logKd/Ki=9.00, IC50=1nM IC50=1nM O14757 21074424 1 FVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKK