3opr A 1.65 BS01 MA4 A 1 V224 P226 I246 A248 V261 A284 E288 V192 P194 I213 A215 V227 A250 E254 S70 K73 S130 K234 A237 S45 K48 S105 K202 A205 3.5.2.6 0008800,0017001,0030655,0046677 P0AD64 21357298 400 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDHALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3opr A 1.65 BS02 MA4 A 2 R244 I279 R211 I245 S70 K73 S130 K234 A237 S45 K48 S105 K202 A205 3.5.2.6 0008800,0017001,0030655,0046677 P0AD64 21357298 401 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDHALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR 3opr A 1.65 BS03 SA2 A 1 S70 Y105 S130 T235 G236 A237 S45 Y80 S105 T203 G204 A205 S70 K73 S130 K234 A237 S45 K48 S105 K202 A205 3.5.2.6 0008800,0017001,0030655,0046677 -logKd/Ki=6.59, Ki=0.26uM P0AD64 21357298 1 SPQPLEQIKLSESQLSGRVGMIEMDLASGRTLTAWRADERFPMMSTFKVVLCGAVLARVDAGDEQLERKIHYRQQDLVDYSPVSEKHLADGMTVGELCAAAITMSDNSAANLLLATVGGPAGLTAFLRQIGDNVTRLDHALPGDARDTTTPASMAATLRKLLTSQRLSARSQRQLLQWMVDDRVAGPLIRSVLPAGWFIADKTGAGERGARGIVALLGPNNKAERIVVIYLRDTPASMAERNQQIAGIGAALIEHWQR