3ook A 2.29 BS01 peptide B 0 V303 K307 E318 I321 L324 K325 P467 L468 E471 I472 V57 K61 E72 I75 L78 K79 P221 L222 E225 I226 ? 0003677,0004879,0006355,0032052,0038183 Q96RI1 21269824 745 ~ 756 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3ook A 2.29 BS02 OOK A 1 I277 L291 M294 H298 M332 F333 R335 S336 I339 F340 I356 M369 Y373 I31 L45 M48 H52 M86 F87 R89 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 -logKd/Ki=8.40, IC50=4nM IC50=4nM, EC50=1400nM Q96RI1 21269824 1 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3ook C 2.29 BS01 peptide D 0 K307 H317 I321 L324 K325 P467 L468 E471 I472 K61 H71 I75 L78 K79 P221 L222 E225 I226 ? 0003677,0004879,0006355,0032052,0038183 Q96RI1 21269824 746 ~ 756 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3ook C 2.29 BS02 OOK C 1 I273 I277 L291 M294 M332 F333 R335 S336 I339 F340 I356 M369 Y373 I27 I31 L45 M48 M86 F87 R89 S90 I93 F94 I110 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 IC50=4nM, EC50=1400nM Q96RI1 21269824 2 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ