3oof A 2.29 BS01 peptide B 0 V303 K307 L324 L468 E471 V57 K61 L78 L222 E225 ? 0003677,0004879,0006355,0032052,0038183 Q96RI1 21269824 745 ~ 756 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3oof A 2.29 BS02 OOF A 1 I277 L291 M294 M332 F333 R335 S336 F340 I356 S359 M369 Y373 I31 L45 M48 M86 F87 R89 S90 F94 I110 S113 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 -logKd/Ki=7.30, IC50=50nM IC50=50nM, EC50=2500nM Q96RI1 21269824 1 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3oof C 2.29 BS01 peptide D 0 K307 H317 E318 I321 L324 P467 L468 E471 K61 H71 E72 I75 L78 P221 L222 E225 ? 0003677,0004879,0006355,0032052,0038183 Q96RI1 21269824 744 ~ 756 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ 3oof C 2.29 BS02 OOF C 1 I273 L291 M294 M332 F333 R335 S336 I339 F340 I356 S359 M369 Y373 I27 L45 M48 M86 F87 R89 S90 I93 F94 I110 S113 M123 Y127 ? 0003677,0004879,0006355,0032052,0038183 IC50=50nM, EC50=2500nM Q96RI1 21269824 2 MELTPDQQTLLHFIMDSYNKQRMPQEITNKILKEAFSAEENFLILTEMATNHVQVLVEFTKKLPGFQTLDHEDQIALLKGSAVEAMFLRSAEIFNKKLPSGHSDLLEARIRNSGISDEYITPMFSFYKSIGELKMTQEEYALLTAIVILSPDRQYIKDREAVEKLQEPLLDVLQKLCKIHQPENPQHFACLLGRLTELRTFNHHHAEMLMSWRVNDHKFTPLLCEIWDVQ