3og7 A 2.45 BS01 032 A 1 I463 A481 L505 L514 T529 W531 C532 F583 D594 F595 G596 I15 A33 L57 L66 T81 W83 C84 F132 D143 F144 G145 D576 K578 N580 N581 D594 S616 D125 K127 N129 N130 D143 S147 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=7.51, IC50=31nM IC50=31nM, Kd=51nM, EC50=2290nM P15056 20823850 1 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTAPQLAIVTQWCEGSSLYHHLHASFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGGSILWMAPEVIRNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELARE