3ndm B 3.3 BS01 3ND B 1 R84 G85 V90 A103 M153 M156 D202 L205 A215 R78 G79 V84 A97 M147 M150 D196 L199 A209 D198 K200 N203 D216 T237 D192 K194 N197 D210 T231 2.7.11.1 0004672,0004674,0005524,0006468 -logKd/Ki=7.96, IC50=11nM Q13464 20471253 900 FETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN 3ndm C 3.3 BS01 3ND C 1 I82 G83 R84 G85 E89 V90 A103 M153 M156 D202 L205 A215 D216 I78 G79 R80 G81 E85 V86 A99 M149 M152 D198 L201 A211 D212 D198 K200 N203 D216 T237 D194 K196 N199 D212 T228 2.7.11.1 0004672,0004674,0005524,0006468 Q13464 20471253 900 MSFETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCTPDYISPEVLKSQGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDISKEAKNLICAFLTDREVLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN 3ndm D 3.3 BS01 3ND D 1 I82 G83 R84 G85 E89 V90 A103 M153 D202 L205 D216 I76 G77 R78 G79 E83 V84 A97 M147 D196 L199 D210 D198 K200 N203 D216 T237 D192 K194 N197 D210 T231 2.7.11.1 0004672,0004674,0005524,0006468 Q13464 20471253 900 FETRFEKMDNLLRDPKSEVNSDCLLDGLDALVYDLDFPALRKNKNIDNFLSRYKDTINKIRDLRMKAEDYEVVKVIGRGAFGEVQLVRHKSTRKVYAMKLLSKFEMIKRSDSAFFWEERDIMAFANSPWVVQLFYAFQDDRYLYMVMEYMPGGDLVNLMSNYDVPEKWARFYTAEVVLALDAIHSMGFIHRDVKPDNMLLDKSGHLKLADFGTCMKMNKEGMVRCDTAVGTPDYISPEVLKSQGGDGYYGRECDWWSVGVFLYEMLVGDTPFYADSLVGTYSKIMNHKNSLTFPDDNDISKEAKNLICAFLTDREVRLGRNGVEEIKRHLFFKNDQWAWETLRDTVAPVVPDLSSDIDTSNFDDLEEDKGEEETFPIPKAFVGNQLPFVGFTYYSN