3nc9 A 2.4 BS01 TR3 B 1 A226 E227 G229 P246 A256 F260 C282 A285 C289 A224 E225 G227 P244 A254 F258 C280 A283 C287 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0016310,0032868,0042802,0042803,0046835,0070061,0070062,0070873 -logKd/Ki=6.48, IC50=330nM IC50=590nM P50053 21033679 299 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3nc9 B 2.4 BS01 TR3 B 2 A226 G229 P246 A256 A229 G232 P249 A259 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0016310,0032868,0042802,0042803,0046835,0070061,0070062,0070873 ic50=330nM -logKd/Ki=6.48, IC50=330nM IC50=590nM P50053 21033679 300 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV