3m11 A 2.75 BS01 AKI A 1 L139 G140 V147 A160 K162 L164 L178 E181 A213 G216 T217 D274 L14 G15 V22 A35 K37 L39 L53 E56 A88 G91 T92 D149 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T157 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=7.37, IC50=43nM IC50=43nM O14965 20550212 1 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSKPS