3lxn A 2.5 BS01 MI1 A 1 L903 G904 E905 G906 G909 V911 A928 K930 I960 E979 Y980 V981 L1030 G1040 D1041 L16 G17 E18 G19 G22 V24 A41 K43 I73 E92 Y93 V94 L143 G153 D154 D1023 A1025 R1027 N1028 D1041 P1064 D136 A138 R140 N141 D154 P174 2.7.10.2 0004672,0004713,0005524,0006468 Ki=4.4nM IC50=489nM, Kd=620nM, Ki=4.39nM P29597 20478313 1 DPTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRDLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYQG