3lxl A 1.74 BS01 IZA A 1 L828 A853 M902 E903 Y904 L905 G908 L956 L15 A40 M89 E90 Y91 L92 G95 L143 D949 A951 R953 N954 D967 D136 A138 R140 N141 D154 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=8.30, IC50=5nM IC50=5nM P52333 20478313 1 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMGVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML