3kvm A 2.0 BS01 FMN A 1 A96 G97 S120 N145 N181 N212 K255 N284 T285 S305 G306 V333 G334 G335 L355 Y356 T357 A66 G67 S90 N115 N151 N182 K225 N254 T255 S275 G276 V303 G304 G305 L325 Y326 T327 G119 N145 F149 S215 N217 T218 K255 N284 G89 N115 F119 S185 N187 T188 K225 N254 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 Q02127 20153645 398 ATGDERFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLPRARFQDSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSPNTAGLRSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRR 3kvm A 2.0 BS02 DOR A 1 N145 Y147 G148 F149 S215 N217 N284 T285 N115 Y117 G118 F119 S185 N187 N254 T255 G119 N145 F149 S215 N217 T218 K255 N284 G89 N115 F119 S185 N187 T188 K225 N254 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 Q02127 20153645 399 ATGDERFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLPRARFQDSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSPNTAGLRSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRR 3kvm A 2.0 BS03 951 A 1 Y38 M43 P52 H56 A59 R136 Y356 T360 P364 Y8 M13 P22 H26 A29 R106 Y326 T330 P334 G119 N145 F149 S215 N217 T218 K255 N284 G89 N115 F119 S185 N187 T188 K225 N254 1.3.5.2 0004151,0004152,0005515,0005654,0005737,0005739,0005743,0005829,0006207,0006221,0006225,0009220,0016020,0016491,0016627,0044205,0106430 ic50=0.5uM Q02127 20153645 402 ATGDERFYAEHLMPTLQGLLDPESAHRLAVRFTSLGLLPRARFQDSDMLEVRVLGHKFRNPVGIAAGFDKHGEAVDGLYKMGFGFVEIGSVTPKPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAKLTEDGLPLGVNLGKNKTSVDAAEDYAEGVRVLGPLADYLVVNVSSPNTAGLRSLQGKAELRRLLTKVLQERDGLRRVHRPAVLVKIAPDLTSQDKEDIASVVKELGIDGLIVTNTTVSRPAGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRVPIIGVGGVSSGQDALEKIRAGASLVQLYTALTFWGPPVVGKVKRELEALLKEQGFGGVTDAIGADHRR