3jsx A 2.45 BS01 FAD A 1 H11 T15 S16 F17 N18 A20 P102 L103 Q104 W105 F106 T147 T148 G149 G150 Y155 I192 R200 H10 T14 S15 F16 N17 A19 P101 L102 Q103 W104 F105 T146 T147 G148 G149 Y154 I191 R199 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx A 2.45 BS02 CC2 A 1 W105 F106 G149 G150 H161 W104 F105 G148 G149 H160 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx A 2.45 BS03 CC2 B 1 Y126 Y128 F178 F232 Y125 Y127 F177 F231 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx B 2.45 BS01 FAD A 1 Q66 P68 Q65 P67 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx B 2.45 BS02 CC2 A 1 Y126 Y128 M131 F232 Y125 Y127 M130 F231 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx B 2.45 BS03 FAD B 1 H11 S16 F17 N18 P102 L103 Q104 W105 F106 T147 T148 G149 G150 Y155 I192 R200 L204 H10 S15 F16 N17 P101 L102 Q103 W104 F105 T146 T147 G148 G149 Y154 I191 R199 L203 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx B 2.45 BS04 CC2 B 1 W105 G150 H161 H194 W104 G149 H160 H193 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx C 2.45 BS01 FAD C 1 H11 F17 N18 A20 P102 L103 Q104 W105 T147 T148 G149 G150 Y155 I192 R200 L204 H10 F16 N17 A19 P101 L102 Q103 W104 T146 T147 G148 G149 Y154 I191 R199 L203 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx C 2.45 BS02 CC2 C 1 W105 G149 G150 M154 H161 H194 W104 G148 G149 M153 H160 H193 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx C 2.45 BS03 CC2 D 1 Y126 Y128 F178 F232 Y125 Y127 F177 F231 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx D 2.45 BS01 CC2 C 1 Y126 Y128 F178 Y125 Y127 F177 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx D 2.45 BS02 FAD D 1 H11 S16 F17 N18 A20 L103 Q104 W105 F106 T147 T148 G149 G150 Y155 I192 R200 H10 S15 F16 N17 A19 L102 Q103 W104 F105 T146 T147 G148 G149 Y154 I191 R199 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx D 2.45 BS03 CC2 D 1 W105 G149 G150 H161 W104 G148 G149 H160 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx E 2.45 BS01 FAD E 1 H11 S16 F17 N18 P102 L103 Q104 W105 F106 T147 T148 G149 Y155 R200 H10 S15 F16 N17 P101 L102 Q103 W104 F105 T146 T147 G148 Y154 R199 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx E 2.45 BS02 CC2 E 1 W105 F106 G149 G150 M154 H161 W104 F105 G148 G149 M153 H160 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx E 2.45 BS03 CC2 G 1 Y126 Y128 M131 F178 Y125 Y127 M130 F177 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx F 2.45 BS01 FAD F 1 H11 S16 F17 N18 A20 L103 Q104 W105 F106 T147 T148 G149 G150 Y155 I192 R200 L204 H10 S15 F16 N17 A19 L102 Q103 W104 F105 T146 T147 G148 G149 Y154 I191 R199 L203 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx F 2.45 BS02 CC2 F 1 W105 G149 G150 M154 H161 W104 G148 G149 M153 H160 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx F 2.45 BS03 FAD H 1 Q66 P68 Q65 P67 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx F 2.45 BS04 CC2 H 1 Y126 Y128 F232 Y125 Y127 F231 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx G 2.45 BS01 CC2 E 1 Y128 M131 F178 F232 Y127 M130 F177 F231 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx G 2.45 BS02 FAD G 1 H11 S16 F17 N18 L103 Q104 W105 F106 T147 T148 G149 Y155 I192 R200 H10 S15 F16 N17 L102 Q103 W104 F105 T146 T147 G148 Y154 I191 R199 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx G 2.45 BS03 CC2 G 1 W105 G149 G150 H161 W104 G148 G149 H160 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx H 2.45 BS01 CC2 F 1 Y126 Y128 F178 Y125 Y127 F177 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx H 2.45 BS02 FAD H 1 H11 S16 F17 N18 P102 L103 Q104 W105 F106 T147 T148 G149 Y155 I192 R200 H10 S15 F16 N17 P101 L102 Q103 W104 F105 T146 T147 G148 Y154 I191 R199 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 P15559 19877692 601 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA 3jsx H 2.45 BS03 CC2 H 1 W105 G149 G150 H161 H194 W104 G148 G149 H160 H193 G149 Y155 H161 G148 Y154 H160 1.6.5.2 0000209,0002931,0003723,0003955,0004128,0004784,0005515,0005634,0005737,0005829,0006116,0006743,0006801,0006805,0006809,0006979,0007271,0007584,0008753,0009410,0009636,0009725,0009743,0014070,0014075,0016491,0019430,0030163,0030425,0032355,0032496,0033574,0034599,0042177,0042360,0042373,0042802,0043025,0043066,0043279,0043525,0045087,0045202,0045454,0045471,0050136,0051602,0070301,0070995,0071248,0110076,1904772,1904844,1904880,1905395 ic50=7.7nM IC50=1095nM P15559 19877692 547 GRRALIVLAHSERTSFNYAMKEAAAAALKKKGWEVVESDLYAMNFNPIISRKDITGKLKDPANFQYPAESVLAYKEGHLSPDIVAEQKKLEAADLVIFQFPLQWFGVPAILKGWFERVFIGEFAYTYAAMYDKGPFRSKKAVLSITTGGSGSMYSLQGIHGDMNVILWPIQSGILHFCGFQVLEPQLTYSIGHTPADARIQILEGWKKRLENIWDETPLYFAPSSLFDLNFQAGFLMKKEVQDEEKNKKFGLSVGHHLGKSIPTDNQIKA