3il5 A 2.6 BS01 B82 A 1 R42 G220 I223 F224 H250 A252 N253 I256 N280 F312 G313 R37 G215 I218 F219 H245 A247 N248 I251 N275 F307 G308 2.3.1.180 0004315,0005737,0006633,0016746,0033818 -logKd/Ki=5.80, IC50=1.6uM IC50=1600nM Q820T1 19665020 401 KNYARISCTSRYVPENCVTNHQLSEMMDTSDEWIHSRTGISERRIVTQENTSDLCHQVAKQLLEKSGKQASEIDFILVATVTPDFNMPSVACQVQGAIGATEAFAFDISAACSGFVYALSMAEKLVLSGRYQTGLVIGGETFSKMLDWTDRSTAVLFGDGAAGVLIEAAETPHFLNEKLQADGQRWAALTSGYTINESPFYQGHKQASKTLQMEGRSIFDFAIKDVSQNILSLVTDETVDYLLLHQANVRIIDKIARKTKISREKFLTNMDKYGNTSAASIPILLDEAVENGTLILGSQQRVVLTGFGGGLTWGSLLLTL 3il5 B 2.6 BS01 B82 B 1 R42 G220 I223 F224 A252 N253 I256 N280 F312 R36 G214 I217 F218 A246 N247 I250 N274 F306 2.3.1.180 0004315,0005737,0006633,0016746,0033818 -logKd/Ki=5.80, IC50=1.6uM IC50=1600nM Q820T1 19665020 401 KNYARISCTSRYVPENCVTNHQLSEMMDTDEWIHSRTGISERRIVTQENTSDLCHQVAKQLLEKSGKQASEIDFILVATVTPDFNMPSVACQVQGAIGATEAFAFDISAACSGFVYALSMAEKLVLSGRYQTGLVIGGETFSKMLDWTDRSTAVLFGDGAAGVLIEAAETPHFLNEKLQADGQRWAALTSGYTINESPFYQGHKQASKTLQMEGRSIFDFAIKDVSQNILSLVTDETVDYLLLHQANVRIIDKIARKTKISREKFLTNMDKYGNTSAASIPILLDEAVENGTLILGSQQRVVLTGFGGGLTWGSLLLTL 3il5 C 2.6 BS01 B82 C 1 R42 G220 I223 F224 H250 A252 N253 R255 I256 N280 F312 G313 R37 G215 I218 F219 H245 A247 N248 R250 I251 N275 F307 G308 2.3.1.180 0004315,0005737,0006633,0016746,0033818 IC50=1600nM Q820T1 19665020 401 KNYARISCTSRYVPENCVTNHQLSEMMDTSDEWIHSRTGISERRIVTQENTSDLCHQVAKQLLEKSGKQASEIDFILVATVTPDFNMPSVACQVQGAIGATEAFAFDISAACSGFVYALSMAEKLVLSGRYQTGLVIGGETFSKMLDWTDRSTAVLFGDGAAGVLIEAAETPHFLNEKLQADGQRWAALTSGYTINESPFYQGHKQASKTLQMEGRSIFDFAIKDVSQNILSLVTDETVDYLLLHQANVRIIDKIARKTKISREKFLTNMDKYGNTSAASIPILLDEAVENGTLILGSQQRVVLTGFGGGLTWGSLLLTL 3il5 D 2.6 BS01 B82 D 1 R42 L161 G220 I223 F224 A252 R255 I256 N280 F312 G313 R37 L156 G215 I218 F219 A247 R250 I251 N275 F307 G308 2.3.1.180 0004315,0005737,0006633,0016746,0033818 IC50=1600nM Q820T1 19665020 401 KNYARISCTSRYVPENCVTNHQLSEMMDTSDEWIHSRTGISERRIVTQENTSDLCHQVAKQLLEKSGKQASEIDFILVATVTPDFNMPSVACQVQGAIGATEAFAFDISAACSGFVYALSMAEKLVLSGRYQTGLVIGGETFSKMLDWTDRSTAVLFGDGAAGVLIEAAETPHFLNEKLQADGQRWAALTSGYTINESPFYQGHKQASKTLQMEGRSIFDFAIKDVSQNILSLVTDETVDYLLLHQANVRIIDKIARKTKISREKFLTNMDKYGNTSAASIPILLDEAVENGTLILGSQQRVVLTGFGGGLTWGSLLLTL