3hyg A 1.4 BS01 ZN A 1 H410 H414 H420 H147 H151 H157 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 901 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg A 1.4 BS02 CA A 1 E270 D353 D360 C471 D474 E7 D90 D97 C208 D211 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 902 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg A 1.4 BS03 CA A 2 E270 D353 D474 E7 D90 D211 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 903 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg A 1.4 BS04 CA A 3 D369 L370 C376 T378 E398 D106 L107 C113 T115 E135 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 904 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg A 1.4 BS05 099 A 1 D377 T378 L379 T407 H410 E411 H414 H420 S440 S441 I442 L443 D114 T115 L116 T144 H147 E148 H151 H157 S177 S178 I179 L180 3.4.24.- 0004222,0006508,0008237 ic50=93nM -logKd/Ki=7.03, IC50=93nM Q9UNA0 19586907 801 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg B 1.4 BS01 ZN B 1 H410 H414 H420 H147 H151 H157 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 901 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg B 1.4 BS02 CA B 1 E270 D353 D360 C471 D474 E7 D90 D97 C208 D211 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 902 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg B 1.4 BS03 CA B 2 E270 D353 D474 E7 D90 D211 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 903 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg B 1.4 BS04 CA B 3 D369 L370 C376 T378 E398 D106 L107 C113 T115 E135 3.4.24.- 0004222,0006508,0008237 Q9UNA0 19586907 904 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI 3hyg B 1.4 BS05 099 B 1 D377 T378 L379 T407 H410 E411 H414 H420 S440 S441 I442 L443 D114 T115 L116 T144 H147 E148 H151 H157 S177 S178 I179 L180 3.4.24.- 0004222,0006508,0008237 ic50=93nM Q9UNA0 19586907 801 SRARQVELLLVADASMARKYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNFCKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHDDSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQI