3gur A 2.5 BS01 BYG A 1 Y6 W7 G11 L12 W45 K49 N58 L59 Q71 S72 R107 A111 Y115 F208 T209 Y6 W7 G11 L12 W45 K49 N58 L59 Q71 S72 R107 A111 Y115 F208 T209 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0004602,0005102,0005504,0005515,0005737,0005829,0006629,0006749,0010880,0010881,0014809,0016529,0016740,0018916,0019899,0042178,0042802,0042803,0043295,0043651,0045171,0051122,0055119,0060315,0060316,0070062,0070458,0071313,0098869 -logKd/Ki=8.00, IC50=0.01uM P28161 19808963 218 PMTLGYWNIRGLAHSIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGTHKITQSNAILRYIARKHNLCGESEKEQIREDILENQFMDSRMQLAKLCYDPDFEKLKPEYLQALPEMLKLYSQFLGKQPWFLGDKITFVDFIAYDVLERNQVFEPSCLDAFPNLKDFISRFEGLEKISAYMKSSRFLPRPVFTKMAVWGNK 3gur B 2.5 BS01 GSH B 1 Y6 W7 L12 R42 W45 K49 N58 L59 Q71 S72 Y6 W7 L12 R42 W45 K49 N58 L59 Q71 S72 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0004602,0005102,0005504,0005515,0005737,0005829,0006629,0006749,0010880,0010881,0014809,0016529,0016740,0018916,0019899,0042178,0042802,0042803,0043295,0043651,0045171,0051122,0055119,0060315,0060316,0070062,0070458,0071313,0098869 P28161 19808963 218 PMTLGYWNIRGLAHSIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGTHKITQSNAILRYIARKHNLCGESEKEQIREDILENQFMDSRMQLAKLCYDPDFEKLKPEYLQALPEMLKLYSQFLGKQPWFLGDKITFVDFIAYDVLERNQVFEPSCLDAFPNLKDFISRFEGLEKISAYMKSSRFLPRPVFTKMAVWGN 3gur C 2.5 BS01 BYG C 1 Y6 W7 G11 L12 R42 W45 N58 L59 Q71 S72 A111 F208 T209 Y6 W7 G11 L12 R42 W45 N58 L59 Q71 S72 A111 F208 T209 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0004602,0005102,0005504,0005515,0005737,0005829,0006629,0006749,0010880,0010881,0014809,0016529,0016740,0018916,0019899,0042178,0042802,0042803,0043295,0043651,0045171,0051122,0055119,0060315,0060316,0070062,0070458,0071313,0098869 P28161 19808963 218 PMTLGYWNIRGLAHSIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGTHKITQSNAILRYIARKHNLCGESEKEQIREDILENQFMDSRMQLAKLCYDPDFEKLKPEYLQALPEMLKLYSQFLGKQPWFLGDKITFVDFIAYDVLERNQVFEPSCLDAFPNLKDFISRFEGLEKISAYMKSSRFLPRPVFTKMAVWGNK 3gur D 2.5 BS01 GSH D 1 Y6 W7 W45 N58 L59 Q71 S72 Y6 W7 W45 N58 L59 Q71 S72 Y6 L12 R17 Y6 L12 R17 2.5.1.18 0004364,0004602,0005102,0005504,0005515,0005737,0005829,0006629,0006749,0010880,0010881,0014809,0016529,0016740,0018916,0019899,0042178,0042802,0042803,0043295,0043651,0045171,0051122,0055119,0060315,0060316,0070062,0070458,0071313,0098869 P28161 19808963 218 PMTLGYWNIRGLAHSIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGTHKITQSNAILRYIARKHNLCGESEKEQIREDILENQFMDSRMQLAKLCYDPDFEKLKPEYLQALPEMLKLYSQFLGKQPWFLGDKITFVDFIAYDVLERNQVFEPSCLDAFPNLKDFISRFEGLEKISAYMKSSRFLPRPVFTKMAVWGNK