3gb2 A 2.4 BS01 G3B A 1 I62 F67 A83 K85 D133 Y134 V135 R141 L188 D200 I28 F33 A49 K51 D94 Y95 V96 R102 L149 D161 D181 K183 N186 D200 S219 D142 K144 N147 D161 S180 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=34nM -logKd/Ki=7.47, IC50=34nM P49841 19775160 999 SKVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHAR