3g1m A 1.7 BS01 RF3 A 1 L87 M102 G106 F110 M142 Y148 T149 N176 N179 E180 L66 M81 G85 F89 M121 Y127 T128 N155 N158 E159 ? 0000976,0003677,0003700,0005515,0005829,0006355,0045892,0046677 ic50=0.522uM -logKd/Ki=6.30, IC50=0.5uM IC50=500nM P9WMC1 19412174 217 GDDRELAILATAENLLEDRPLADISVDDLAKGAGISRPTFYFYFPSKEAVLLTLLDRVVNQADMALQTLAENPADTDRENMWRTGINVFFETFGSHKAVTRAGQAARATSVEVAELWSTFMQKWIAYTAAVIDAERDRGAAPRTLPAHELATALNLMNERTLFASFAGEQPSVPEARVLDTLVHIWVTSIYGEN