3fr0 A 2.7 BS01 GLC A 1 S151 F152 T168 K169 N204 D205 N231 E256 E290 S138 F139 T155 K156 N191 D192 N218 E243 E277 R85 S151 N166 D205 R72 S138 N153 D192 2.7.1.1 0001678,0004340,0004396,0005515,0005524,0005536,0005634,0005654,0005737,0005739,0005829,0005975,0006006,0006007,0006096,0006110,0006739,0008865,0009749,0016301,0016310,0016773,0019158,0019318,0032024,0032869,0042593,0043266,0044320,0045721,0045725,0046835,0050796,0051156,0061621,0070509,0141089,1901135 P35557 19188063 500 TLVEQILAEFQLQEEDLKKVMRRMQKEMDRGLRLETHEEASVKMLPTYVRSTPEGSEVGDFLSLDLGGTNFRVMLVKVGEGEEGQWSVKTKHQMYSIPEDAMTGTAEMLFDYISECISDFLDKHQMKHKKLPLGFTFSFPVRHEDIDKGILLNWTKGFKASGAEGNNVVGLLRDAIKRRGDFEMDVVAMVNDTVATMISCYYEDHQCEVGMIVGTGCNACYMEEMQNVELVEGDEGRMCVNTEWGAFGDSGELDEFLLEYDRLVDESSANPGQQLYEKLIGGKYMGELVRLVLLRLVDENLLFHGEASEQLRTRGAFETRFVSQVESDTGDRKQIYNILSTLGLRPSTTDCDIVRRACESVSTRAAHMCSAGLAGVINRMRESRSEDVMRITVGVDGSVYKLHPSFKERFHASVRRLTPSCEITFIESEEGSGRGAALVSAVACKKAC 3fr0 A 2.7 BS02 AJB A 1 Y61 V62 R63 S64 I211 Y214 Y215 M235 V452 V455 Y48 V49 R50 S51 I198 Y201 Y202 M222 V439 V442 R85 S151 N166 D205 R72 S138 N153 D192 2.7.1.1 0001678,0004340,0004396,0005515,0005524,0005536,0005634,0005654,0005737,0005739,0005829,0005975,0006006,0006007,0006096,0006110,0006739,0008865,0009749,0016301,0016310,0016773,0019158,0019318,0032024,0032869,0042593,0043266,0044320,0045721,0045725,0046835,0050796,0051156,0061621,0070509,0141089,1901135 EC50=420nM, Kd=440nM P35557 19188063 501 TLVEQILAEFQLQEEDLKKVMRRMQKEMDRGLRLETHEEASVKMLPTYVRSTPEGSEVGDFLSLDLGGTNFRVMLVKVGEGEEGQWSVKTKHQMYSIPEDAMTGTAEMLFDYISECISDFLDKHQMKHKKLPLGFTFSFPVRHEDIDKGILLNWTKGFKASGAEGNNVVGLLRDAIKRRGDFEMDVVAMVNDTVATMISCYYEDHQCEVGMIVGTGCNACYMEEMQNVELVEGDEGRMCVNTEWGAFGDSGELDEFLLEYDRLVDESSANPGQQLYEKLIGGKYMGELVRLVLLRLVDENLLFHGEASEQLRTRGAFETRFVSQVESDTGDRKQIYNILSTLGLRPSTTDCDIVRRACESVSTRAAHMCSAGLAGVINRMRESRSEDVMRITVGVDGSVYKLHPSFKERFHASVRRLTPSCEITFIESEEGSGRGAALVSAVACKKAC