3fqe A 2.5 BS01 P5C A 1 L377 S379 V385 A400 M448 G454 P455 R498 L501 S511 D512 L15 S17 V23 A38 M81 G87 P88 R131 L134 S144 D145 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K163 2.7.10.2 0004672,0004713,0005524,0006468 Ki~0.0125uM -logKd/Ki=8.30, Ki=5nM IC50=4nM, EC50=2500nM P43405 19220318 1 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH