3fhr A 1.9 BS01 P4O A 1 L50 L52 G53 V58 A71 K73 M121 E122 L173 T186 D187 L18 L20 G21 V26 A39 K41 M89 E90 L140 T153 D154 D166 K168 N171 D187 D133 K135 N138 D154 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=6.68, IC50=210nM IC50=210nM Q16644 19937655 1 EPKKYAVTDDYQLSKQVLGLGVNGKVLECFHRRTGQKCALKLLYDSPKARQEVDHHWQASGGPHIVCILDVYENMHHGKRCLLIIMECMEGGELFSRIQERDQAFTEREAAEIMRDIGTAIQFLHSHNIAHRDVKPENLLYTSKEKDAVLKLTDFGFAKETEKYDKSCDMWSLGVIMYILLCGFPPFGFPNPEWSEVSEDAKQLIRLLLKTDPTERLTITQFMNHPWINQSMVVPQTPLHTARVLQEDKDHWDEVKEEMTSALATMRVDYDQV