3f3w A 2.6 BS01 1BU A 1 A293 E310 M314 M341 L393 A403 D404 F405 A37 E54 M58 M85 L137 A147 D148 F149 D386 R388 A390 N391 D404 F424 D130 R132 A134 N135 D148 F152 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=7.47, IC50=34nM IC50=21nM, Kd=73nM P00523 19462975 1 KDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3f3w B 2.6 BS01 1BU B 1 L273 A293 E310 M314 V323 Y340 M341 A403 D404 F405 L16 A36 E53 M57 V66 Y83 M84 A146 D147 F148 D386 R388 A390 N391 D404 F424 D129 R131 A133 N134 D147 F151 2.7.10.2 0004672,0004713,0005524,0006468 IC50=21nM, Kd=73nM P00523 19462975 1 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVMEYMSKGCLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL