3eb1 A 2.4 BS01 LZQ A 1 Y46 D48 A217 G220 Q262 Q266 Y45 D47 A216 G219 Q261 Q265 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=16.3uM -logKd/Ki=4.79, Ki=16.3uM IC50=20000nM P18031 19012396 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGD