3e8r A 1.9 BS01 ZN A 1 H405 H409 H415 H184 H188 H194 3.4.24.86 0004222,0006508,0008237 P78536 18835710 1 PDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3e8r A 1.9 BS02 615 A 1 T347 L348 G349 E398 L401 H405 E406 H409 H415 Y433 V434 P437 A439 T130 L131 G132 E177 L180 H184 E185 H188 H194 Y212 V213 P216 A218 3.4.24.86 0004222,0006508,0008237 -logKd/Ki=9.74, Ki=0.18nM Ki=0.180000nM P78536 18835710 486 PDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3e8r A 1.9 BS03 INN A 1 M345 G346 T347 Y390 H405 E406 H409 H415 P437 I438 A439 M128 G129 T130 Y169 H184 E185 H188 H194 P216 I217 A218 3.4.24.86 0004222,0006508,0008237 P78536 18835710 4 PDPMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAGDHENNKMFSQCSKQSIYKTIESKAQECFQERS 3e8r B 1.9 BS01 ZN B 1 H405 H409 H415 H186 H190 H196 3.4.24.86 0004222,0006508,0008237 P78536 18835710 2 PMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQER 3e8r B 1.9 BS02 615 B 1 T347 L348 G349 E398 L401 H405 E406 H409 H415 Y433 V434 Y436 P437 A439 V440 G442 N447 T128 L129 G130 E179 L182 H186 E187 H190 H196 Y214 V215 Y217 P218 A220 V221 G223 N228 3.4.24.86 0004222,0006508,0008237 Ki=0.180000nM P78536 18835710 486 PMKNTCKLLVVADHRFYRYMGRGEESTTTNYLIELIDRVDDIYRNTAWDNAGFKGYGIQIEQIRILKSPQEVKPGEKHYNMAKSYPNEEKDAWDVKMLLEQFSFDIAEEASKVCLAHLFTYQDFDMGTLGLAYGGSPRANSHGGVCPKAYYSPVGKKNIYLNSGLTSTKNYGKTILTKEADLVTTHELGHNFGAEHDPDGLAECAPNEDQGGKYVMYPIAVSGDHENNKMFSQCSKQSIYKTIESKAQECFQER