3dng A 2.0 BS01 CA A 1 D137 G169 G171 D173 D58 G90 G92 D94 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 996 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng A 2.0 BS02 CA A 2 D154 G155 N157 I159 D177 E180 D75 G76 N78 I80 D98 E101 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 997 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng A 2.0 BS03 ZN A 1 H147 D149 H162 H175 H68 D70 H83 H96 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 998 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng A 2.0 BS04 ZN A 2 H197 H201 H207 H118 H122 H128 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 999 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng A 2.0 BS05 AXA A 1 L193 H197 L214 Y216 P217 N218 Y219 A220 F221 R222 Y227 P230 L114 H118 L135 Y137 P138 N139 Y140 A141 F142 R143 Y148 P151 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=7.4nM -logKd/Ki=8.13, IC50=7.4nM IC50=7.4nM P22894 19173605 1 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng B 2.0 BS01 CA B 1 D137 G169 G171 D173 D58 G90 G92 D94 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 996 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng B 2.0 BS02 CA B 2 D154 G155 N157 I159 D177 E180 D75 G76 N78 I80 D98 E101 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 997 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng B 2.0 BS03 ZN B 1 H147 D149 H162 H175 H68 D70 H83 H96 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 998 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng B 2.0 BS04 ZN B 2 H197 H201 H207 H118 H122 H128 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 P22894 19173605 999 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG 3dng B 2.0 BS05 AXA B 1 L193 H197 L214 Y216 P217 N218 Y219 A220 F221 R222 Y227 P230 L114 H118 L135 Y137 P138 N139 Y140 A141 F142 R143 Y148 P151 H197 E198 H201 H207 H118 E119 H122 H128 3.4.24.34 0004222,0006508,0008237,0008270,0031012 ic50=7.4nM IC50=7.4nM P22894 19173605 2 MLTPGNPKWERTNLTYRIRNYTPQLSEAEVERAIKDAFELWSVASPLIFTRISQGEADINIAFYQRDHGDNSPFDGPNGILAHAFQPGQGIGGDAHFDAEETWTNTSANYNLFLVAAHEFGHSLGLAHSSDPGALMYPNYAFRETSNYSLPQDDIDGIQAIYG