3d4q A 2.8 BS01 SM5 A 1 I463 G464 S465 V471 A481 K483 E501 W531 C532 F583 D594 I16 G17 S18 V24 A34 K36 E54 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S157 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=10.52, IC50=0.03nM IC50=0.030000nM P15056 18676143 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK 3d4q B 2.8 BS01 SM5 B 1 I463 G464 S465 V471 A481 K483 E501 W531 C532 F583 D594 I16 G17 S18 V24 A34 K36 E54 W84 C85 F136 D147 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S157 2.7.11.1 0004672,0005524,0006468 IC50=0.030000nM P15056 18676143 1 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK