3cpc A 2.4 BS01 C52 A 1 V848 A866 K868 E885 L889 V899 T916 C919 L1035 C1045 D1046 F1047 V23 A41 K43 E60 L64 V74 T91 C94 L160 C170 D171 F172 D1028 A1030 R1032 N1033 D1046 D153 A155 R157 N158 D171 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 -logKd/Ki=5.30, IC50=5uM IC50=>5000nM P35968 18447379 1 LPYDASKWEFPRDRLKLGKPLQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 3cpc B 2.4 BS01 C52 B 1 V848 A866 K868 E885 V899 T916 C919 L1035 I1044 C1045 D1046 F1047 V24 A42 K44 E58 V72 T89 C92 L150 I159 C160 D161 F162 D1028 A1030 R1032 N1033 D1046 D143 A145 R147 N148 D161 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 IC50=>5000nM P35968 18447379 2 LPYDASKWEFPRDRLKLGKPLGQVIEADAFGIDKTATCRTVAVKMLATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQ