3cp9 A 2.5 BS01 C19 A 1 L840 V848 A866 K868 E885 L889 V898 T916 C919 L1035 C1045 D1046 F1047 L24 V26 A44 K46 E63 L67 V76 T94 C97 L163 C173 D174 F175 D1028 A1030 R1032 N1033 D1046 D156 A158 R160 N161 D174 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 -logKd/Ki=7.32, IC50=0.048uM IC50=48nM P35968 18447379 501 AERLPYDASKWEFPRDRLKLGKPLQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHHHHH 3cp9 B 2.5 BS01 C19 B 1 V848 A866 K868 E885 L889 V898 T916 C919 L1035 C1045 D1046 F1047 V28 A46 K48 E62 L66 V75 T93 C96 L156 C166 D167 F168 D1028 A1030 R1032 N1033 D1046 D149 A151 R153 N154 D167 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 IC50=48nM P35968 18447379 502 RLPYDASKWEFPRDRLKLGKPLGRGGQVIEADAFGIDKTATCRTVAVKMLATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQ