3bmq A 1.7 BS01 NAP A 1 R14 I15 Y34 H35 N36 S37 L63 N93 A94 S95 T126 L159 K178 P204 G205 S207 L208 R13 I14 Y33 H34 N35 S36 L62 N92 A93 S94 T117 L144 K163 P189 G190 S192 L193 R14 D161 Y174 K178 R13 D146 Y159 K163 ? 0000166,0016491,0047040 O76290 19916554 269 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQKGSSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq A 1.7 BS02 AX5 A 1 S95 F97 Y174 L208 P210 M213 S94 F96 Y159 L193 P195 M198 R14 D161 Y174 K178 R13 D146 Y159 K163 ? 0000166,0016491,0047040 Ki=3.2uM -logKd/Ki=5.49, Ki=3.2uM O76290 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQKGSSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq B 1.7 BS01 NAP B 1 R14 I15 Y34 H35 N36 S37 L63 N93 A94 S95 T126 L159 K178 P204 G205 S207 R13 I14 Y33 H34 N35 S36 L62 N92 A93 S94 T118 L143 K162 P188 G189 S191 R14 D161 Y174 K178 R13 D145 Y158 K162 ? 0000166,0016491,0047040 O76290 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQNGKTVETQVAELIGTNAIAPFLLTMSFAQRQKSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq B 1.7 BS02 AX5 B 1 R14 S95 F97 Y174 P210 R13 S94 F96 Y158 P194 R14 D161 Y174 K178 R13 D145 Y158 K162 ? 0000166,0016491,0047040 Ki=3.2uM O76290 19916554 271 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQNGKTVETQVAELIGTNAIAPFLLTMSFAQRQKSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq C 1.7 BS01 NAP C 1 R14 I15 H33 Y34 H35 N36 S37 D62 L63 N93 A94 S95 T126 L159 K178 P204 G205 S207 R13 I14 H32 Y33 H34 N35 S36 D61 L62 N92 A93 S94 T118 L142 K161 P187 G188 S190 R14 D161 Y174 K178 R13 D144 Y157 K161 ? 0000166,0016491,0047040 O76290 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq C 1.7 BS02 AX5 C 1 S95 F97 Y174 P210 W221 S94 F96 Y157 P193 W204 R14 D161 Y174 K178 R13 D144 Y157 K161 ? 0000166,0016491,0047040 Ki=3.2uM O76290 19916554 271 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq D 1.7 BS01 NAP D 1 R14 I15 Y34 H35 N36 S37 L63 N93 A94 S95 T126 L159 K178 P204 G205 S207 R13 I14 Y33 H34 N35 S36 L62 N92 A93 S94 T117 L144 K163 P189 G190 S192 R14 D161 Y174 K178 R13 D146 Y159 K163 ? 0000166,0016491,0047040 O76290 19916554 269 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQKGSSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3bmq D 1.7 BS02 AX5 D 1 S95 F97 Y174 L208 L209 P210 S94 F96 Y159 L193 L194 P195 R14 D161 Y174 K178 R13 D146 Y159 K163 ? 0000166,0016491,0047040 Ki=3.2uM O76290 19916554 270 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVQGKTVETQVAELIGTNAIAPFLLTMSFAQRQKGSSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA