3bbb B 1.3 BS01 DG B 1 F60 L64 T94 F59 L63 T93 K12 Y52 N115 H118 E129 K11 Y51 N114 H117 E128 2.7.13.3,2.7.4.6 0001726,0003677,0003713,0004550,0004673,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0016310,0018106,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 P22392 19435876 153 ANLERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbb C 1.3 BS01 DA C 1 K12 Y52 V112 K8 Y48 V108 K12 Y52 N115 H118 E129 K8 Y48 N111 H114 E125 2.7.13.3,2.7.4.6 0001726,0003677,0003713,0004550,0004673,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0016310,0018106,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 -logKd/Ki=7.00, Kd=100nM P22392 19435876 153 ERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbb C 1.3 BS02 DG C 1 L55 F60 L64 T94 L51 F56 L60 T90 K12 Y52 N115 H118 E129 K8 Y48 N111 H114 E125 2.7.13.3,2.7.4.6 0001726,0003677,0003713,0004550,0004673,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0016310,0018106,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 -logKd/Ki=7.00, Kd=100nM P22392 19435876 154 ERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbb E 1.3 BS01 DA E 1 Y52 V112 Y48 V108 K12 Y52 N115 H118 E129 K8 Y48 N111 H114 E125 2.7.13.3,2.7.4.6 0001726,0003677,0003713,0004550,0004673,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0016310,0018106,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 P22392 19435876 153 ERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbb E 1.3 BS02 DG E 1 F60 T94 F56 T90 K12 Y52 N115 H118 E129 K8 Y48 N111 H114 E125 2.7.13.3,2.7.4.6 0001726,0003677,0003713,0004550,0004673,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0016310,0018106,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 P22392 19435876 154 ERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE 3bbb F 1.3 BS01 DG F 1 K12 Y52 L55 F60 L64 V112 G113 K11 Y51 L54 F59 L63 V111 G112 K12 Y52 N115 H118 E129 K11 Y51 N114 H117 E128 2.7.13.3,2.7.4.6 0001726,0003677,0003713,0004550,0004673,0005515,0005524,0005576,0005634,0005737,0005829,0005925,0006183,0006228,0006241,0007155,0007229,0009117,0009142,0016301,0016310,0018106,0019003,0030027,0034774,0042802,0042981,0042995,0043066,0045618,0045682,0045893,0045944,0046872,0048471,0050679,0051880,0070062,0071944,1904813 P22392 19435876 153 ANLERTFIAIKPDGVQRGLVGEIIKRFEQKGFRLVAMKFLRASEEHLKQHYIDLKDRPFFPGLVKYMNSGPVVAMVWEGLNVVKTGRVMLGETNPADSKPGTIRGDFCIQVGRNIIHGSDSVKSAEKEISLWFKPEELVDYKSCAHDWVYE